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Cat. No. Product Name Target Signaling Pathways
T16161 Mutant IDH1 inhibitor

Dehydrogenase; Isocitrate Dehydrogenase (IDH) Metabolism
Mutant IDH1 inhibitor 是一种突变型IDH1 R132H 的抑制剂,IC50<72 nM。
T12128 Mutant IDH1-IN-2

Isocitrate Dehydrogenase (IDH) Metabolism
Mutant IDH1-IN-2是突变型异柠檬酸脱氢酶蛋白抑制剂, 在荧光生物化学检测中IC50为16.6 nM,LS-MS 生物化学检测中IC50为<22 nM,。
T2043 Mutant IDH1-IN-1

IDH1-IN-1

Dehydrogenase; Isocitrate Dehydrogenase (IDH) Metabolism
Mutant IDH1-IN-1IDH1突变体的选择性抑制剂,能够作用于突变体 IDH1 R132C/R132C (IC50:4 nM) ,IDH1 R132H/R132H (IC50:42 nM) ,IDH1 R132H/WT (IC50:80 nM) 和野生型 IDH1 (IC50:143 nM)。
T7741 DS-1001b

Dehydrogenase; Isocitrate Dehydrogenase (IDH) Metabolism
DS-1001b 是IDH-1(异柠檬酸脱氢酶-1) 突变体抑制剂。
T7307 Vorasidenib

PVM/MA,PVM/MA共聚物,AG-881

Isocitrate Dehydrogenase (IDH) Metabolism
Vorasidenib (PVM/MA) 是口服具有活力的、脑渗透的突变体异柠檬酸脱氢酶 1 和 2 双重抑制剂。
T16384 Olutasidenib

FT-2102

Dehydrogenase; Isocitrate Dehydrogenase (IDH) Metabolism
Olutasidenib (FT-2102) 是一种可透过血脑屏障的、具有口服活性的、突变型异柠檬酸脱氢酶(IDH)1的选择性有效抑制剂,对IDH1- R132H 和 IDH1- R132C 的IC50分别为 21.2 nM 和 114 nM,可用于急性髓性白血病或骨髓增生异常综合征的研究。
T12129 Mutant IDH1-IN-4

Others Others
Mutant IDH1-IN-4 is an mutant Isocitrate dehydrogenase 1 (IDH 1) inhibitor.

化合物

Mutant IDH1 inhibitor
Cat.No: T16161
Synonym:
Target: Dehydrogenase, Isocitrate Dehydrogenase (IDH)
Mutant IDH1-IN-2
Cat.No: T12128
Synonym:
Target: Isocitrate Dehydrogenase (IDH)
Mutant IDH1-IN-1
Cat.No: T2043
Synonym: IDH1-IN-1
Target: Dehydrogenase, Isocitrate Dehydrogenase (IDH)
DS-1001b
Cat.No: T7741
Synonym:
Target: Dehydrogenase, Isocitrate Dehydrogenase (IDH)
Vorasidenib
Cat.No: T7307
Synonym: PVM/MA,PVM/MA共聚物,AG-881
Target: Isocitrate Dehydrogenase (IDH)
Olutasidenib
Cat.No: T16384
Synonym: FT-2102
Target: Dehydrogenase, Isocitrate Dehydrogenase (IDH)
Mutant IDH1-IN-4
Cat.No: T12129
Synonym:
Target: Others
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